Quotient Sciences Quotient Sciences

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            CMS will be responsible for the development and commercialization of INCB54707 (povorcitinib), a selective oral JAK1 inhibitor, which is being evaluated for non-segmental vitiligo, hidradenitis suppurativa, prurigo nodularis, asthma & chronic spontaneous urticaria.

            Lead Product(s): Povorcitinib

            Therapeutic Area: Dermatology Product Name: INCB054707

            Highest Development Status: Phase III Product Type: Small molecule

            Partner/Sponsor/Collaborator: China Medical System Holdings Limited

            Deal Size: Undisclosed Upfront Cash: Undisclosed

            Deal Type: Licensing Agreement April 01, 2024

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            INCB54707 (povorcitinib) is an oral small-molecule JAK1 inhibitor currently in Phase 2 clinical trials for adult patients with prurigo nodularis. A Phase 3 trial is being planned for prurigo nodularis.

            Lead Product(s): Povorcitinib

            Therapeutic Area: Dermatology Product Name: INCB054707

            Highest Development Status: Phase II Product Type: Small molecule

            Partner/Sponsor/Collaborator: Not Applicable

            Deal Size: Not Applicable Upfront Cash: Not Applicable

            Deal Type: Not Applicable March 10, 2024

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            Opzelura (ruxolitinib phosphate), a novel topical cream formulation with selective JAK1/JAK2 inhibitor, is in phase 2 trial for the treatment of adults with Hurley stage 1 or 2 (mild-to-moderate) hidradenitis suppurativa.

            Lead Product(s): Ruxolitinib Phosphate

            Therapeutic Area: Dermatology Product Name: Opzelura

            Highest Development Status: Phase II Product Type: Small molecule

            Partner/Sponsor/Collaborator: Not Applicable

            Deal Size: Not Applicable Upfront Cash: Not Applicable

            Deal Type: Not Applicable March 10, 2024

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            INCA034176 (axatilimab) is an investigational monoclonal antibody that targets CSF-1R. It is bein evaluated for the treatment of chronic graft-versus-host disease.

            Lead Product(s): Axatilimab

            Therapeutic Area: Immunology Product Name: INCA034176

            Highest Development Status: Phase III Product Type: Large molecule

            Partner/Sponsor/Collaborator: Syndax Pharmaceuticals

            Deal Size: Not Applicable Upfront Cash: Not Applicable

            Deal Type: Not Applicable February 27, 2024

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            Under the agreement, Incyte gains exclusive global rights for tafasitamab, a humanized Fc-modified CD19-targeting immunotherapy marketed in the U.S. as Monjuvi (tafasitamab-cxix) and outside of the U.S. as Minjuvi (tafasitamab).

            Lead Product(s): Tafasitamab

            Therapeutic Area: Oncology Product Name: Monjuvi

            Highest Development Status: Approved Product Type: Large molecule

            Recipient: MorphoSys

            Deal Size: $25.0 million Upfront Cash: Undisclosed

            Deal Type: Agreement February 05, 2024

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            Under the collaboration, AbCellera and Incyte will discover and develop therapeutic antibodies in oncology and Incyte will have the right to develop and commercialize therapeutic antibodies resulting from the collaboration.

            Lead Product(s): Undisclosed

            Therapeutic Area: Oncology Product Name: Undisclosed

            Highest Development Status: Discovery Product Type: Large molecule

            Recipient: AbCellera

            Deal Size: Undisclosed Upfront Cash: Undisclosed

            Deal Type: Collaboration September 13, 2023

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            Syros used its proprietary gene control platform to identify novel therapeutic targets with a focus in myeloproliferative neoplasms, and Incyte received options to obtain worldwide rights to intellectual property resulting from the collaboration for up to 7 validated targets.

            Lead Product(s): Undisclosed

            Therapeutic Area: Oncology Product Name: Undisclosed

            Highest Development Status: Discovery Product Type: Undisclosed

            Recipient: Syros Pharmaceuticals

            Deal Size: $189.0 million Upfront Cash: $10.0 million

            Deal Type: Termination August 14, 2023

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            The collaboration aims to study RP1, Replimune’s lead product candidate, in combination with INCB99280, Incyte’s small molecule oral PD-L1 inhibitor, in patients with high risk, resectable cutaneous squamous cell carcinoma.

            Lead Product(s): Vusolimogene Oderparepvec,INCB99280

            Therapeutic Area: Oncology Product Name: RP1

            Highest Development Status: Preclinical Product Type: Large molecule

            Recipient: Replimune

            Deal Size: Undisclosed Upfront Cash: Undisclosed

            Deal Type: Collaboration July 31, 2023

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            Results showed that patients with AD treated with Opzelura (ruxolitinib) experienced a rapid and substantial improvement in itch, which was sustained and further improved through 28 days of treatment in patients with atopic dermatitis.

            Lead Product(s): Ruxolitinib Phosphate

            Therapeutic Area: Dermatology Product Name: Opzelura

            Highest Development Status: Approved Product Type: Small molecule

            Partner/Sponsor/Collaborator: Not Applicable

            Deal Size: Not Applicable Upfront Cash: Not Applicable

            Deal Type: Not Applicable July 11, 2023

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            Opzelura (ruxolitinib phosphate), a novel cream formulation, is the first and only topical JAK inhibitor approved for use in the UK indicated for the treatment of non-segmental vitiligo with facial involvement in adults and adolescents from 12 years of age.

            Lead Product(s): Ruxolitinib Phosphate

            Therapeutic Area: Dermatology Product Name: Opzelura

            Highest Development Status: Approved Product Type: Small molecule

            Partner/Sponsor/Collaborator: Not Applicable

            Deal Size: Not Applicable Upfront Cash: Not Applicable

            Deal Type: Not Applicable July 05, 2023

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