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01 2Alcon Canada Inc.

02 2Gowling WLG (Canada) LLP

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PharmaCompass

01

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SCI Medicinal Chemistry
Not Confirmed
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SCI Medicinal Chemistry
Not Confirmed

Brinzolamide, Timolol Maleate

Brand Name : AZARGA

Patent Number : 2080223

Filing Date : 1991-04-03

Strength per Unit : 1% / 0.5%

Dosage Form : suspension

Human Or VET : Human

Route of Administration : ophthalmic (topical)

Patent Expiration Date : 2011-04-03

Date Granted : 2000-11-07

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02

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SCI Medicinal Chemistry
Not Confirmed
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SCI Medicinal Chemistry
Not Confirmed

Brinzolamide, Timolol Maleate

Brand Name : AZARGA

Patent Number : 2310230

Filing Date : 1998-11-05

Strength per Unit : 1% / 0.5%

Dosage Form : suspension

Human Or VET : Human

Route of Administration : ophthalmic (topical)

Patent Expiration Date : 2018-11-05

Date Granted : 2008-05-06

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03

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SCI Medicinal Chemistry
Not Confirmed
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SCI Medicinal Chemistry
Not Confirmed

Brinzolamide

Brand Name : AZOPT

Patent Number : 2080223

Filing Date : 1991-04-03

Strength per Unit : 10mg/ml

Dosage Form : Suspension

Human Or VET : Human

Route of Administration : Topical (Ophthalmic)

Patent Expiration Date : 2011-04-03

Date Granted : 2000-11-07

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04

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SCI Medicinal Chemistry
Not Confirmed
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SCI Medicinal Chemistry
Not Confirmed

BRIMONIDINE TARTRATE, BRINZOLAMIDE

Brand Name : SIMBRINZA

Patent Number : 2763778

Filing Date : 2010-06-17

Strength per Unit : 1.0% / 0.2% w / v

Dosage Form : SUSPENSION

Human Or VET : Human

Route of Administration : OPHTHALMIC

Patent Expiration Date : 2030-06-17

Date Granted : 2016-02-02

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