Find Pentazocine manufacturers, exporters & distributors on PharmaCompass

PharmaCompass

Synopsis

ACTIVE PHARMA INGREDIENTS

0

CEP/COS

CEP/COS Certifications

0

EU WC

EU WC

0

KDMF

KDMF

0

VMF

NDC API

API REF. PRICE (USD/KG)

MARKET PLACE

0 DRUGS IN DEVELOPMENT

FDF Dossiers

DRUG PRODUCT COMPOSITIONS

REF. STANDARDS OR IMPURITIES

0

EDQM

0

JP

PATENTS & EXCLUSIVITIES

0

US Patents

0

US Exclusivities

0

Health Canada Patents

DIGITAL CONTENT

0

Data Compilation #PharmaFlow

0

Stock Recap #PipelineProspector

0

Weekly News Recap #Phispers

0

News #PharmaBuzz

GLOBAL SALES INFORMATION

US Medicaid

NA

Annual Reports

NA

115 RELATED EXCIPIENT COMPANIES

207EXCIPIENTS BY APPLICATIONS

Chemistry

Click the arrow to open the dropdown
read-moreClick the button for full data set
Also known as: 17146-95-1, Pentazocine lactate [usan], 1p2xib510o, (1r,9r,13r)-1,13-dimethyl-10-(3-methylbut-2-enyl)-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol;2-hydroxypropanoic acid, (2r*,6r*,11r*)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocin-8-ol lactate (salt), Talwin (lactate)
Molecular Formula
C22H33NO4
Molecular Weight
375.5  g/mol
InChI Key
QNLDTXPVZPRSAM-DTOXXUQYSA-N
FDA UNII
1P2XIB510O

Pentazocine
The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)
1 2D Structure

Pentazocine

2 Identification
2.1 Computed Descriptors
2.1.1 IUPAC Name
(1R,9R,13R)-1,13-dimethyl-10-(3-methylbut-2-enyl)-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol;2-hydroxypropanoic acid
2.1.2 InChI
InChI=1S/C19H27NO.C3H6O3/c1-13(2)7-9-20-10-8-19(4)14(3)18(20)11-15-5-6-16(21)12-17(15)19;1-2(4)3(5)6/h5-7,12,14,18,21H,8-11H2,1-4H3;2,4H,1H3,(H,5,6)/t14-,18+,19+;/m0./s1
2.1.3 InChI Key
QNLDTXPVZPRSAM-DTOXXUQYSA-N
2.1.4 Canonical SMILES
CC1C2CC3=C(C1(CCN2CC=C(C)C)C)C=C(C=C3)O.CC(C(=O)O)O
2.1.5 Isomeric SMILES
C[C@H]1[C@H]2CC3=C([C@@]1(CCN2CC=C(C)C)C)C=C(C=C3)O.CC(C(=O)O)O
2.2 Other Identifiers
2.2.1 UNII
1P2XIB510O
2.3 Synonyms
2.3.1 MeSH Synonyms

1. Fortral

2. Hydrochloride, Pentazocine

3. Lactate, Pentazocine

4. Lexir

5. Pentazocine

6. Pentazocine Hydrochloride

7. Talwin

2.3.2 Depositor-Supplied Synonyms

1. 17146-95-1

2. Pentazocine Lactate [usan]

3. 1p2xib510o

4. (1r,9r,13r)-1,13-dimethyl-10-(3-methylbut-2-enyl)-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol;2-hydroxypropanoic Acid

5. (2r*,6r*,11r*)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocin-8-ol Lactate (salt)

6. Talwin (lactate)

7. Pentalgine

8. Talwin (as Lactate)

9. Unii-1p2xib510o

10. Talwin Injection

11. Einecs 241-209-9

12. Einecs 304-943-1

13. Talwin (tn)

14. Pentazocine Lactate (usp)

15. Schembl42094

16. (all-r)-pentazocine Dl-lactate

17. Chembl1200327

18. Pentazocine Lactate [mi]

19. Dtxsid101027503

20. Pentazocine Lactate [vandf]

21. Pentazocine Lactate [mart.]

22. Pentazocine Lactate [who-dd]

23. Pentazocine Lactate [green Book]

24. Pentazocine Lactate [orange Book]

25. 2-hydroxypropanoic Acid Compd. With (2alpha,6alpha,11r*)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-2,6-methanol-3-benzocin-8-ol (1:1)

26. Lactic Acid, Compd. With 1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocin-8-ol (1:1)

27. Lactic Acid, Compound With (2alpha,6alpha,11r*)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methylbut-2-enyl)-2,6-methano-3-benzocin-8-ol (1:1)

28. Pentazocine Lactate [ep Monograph]

29. D02111

30. Q27252701

31. 2,6-methano-3-benzazocin-8-ol, 1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-, (2.alpha.,6.alpha.,11r*)-, Compd. With 2-hydroxypropanoic Acid (1:1)

32. 2,6-methano-3-benzazocin-8-ol, 1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-, (2alpha,6alpha,11r*)-, Compd. With 2-hydroxypropanoic Acid (1:1)

33. Propanoic Acid, 2-hydroxy-, Compd. With (2alpha,6alpha,11r*)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-2,6-methanol-3-benzocin-8-ol (1:1)

2.4 Create Date
2005-06-24
3 Chemical and Physical Properties
Molecular Weight 375.5 g/mol
Molecular Formula C22H33NO4
Hydrogen Bond Donor Count3
Hydrogen Bond Acceptor Count5
Rotatable Bond Count3
Exact Mass375.24095853 g/mol
Monoisotopic Mass375.24095853 g/mol
Topological Polar Surface Area81 Ų
Heavy Atom Count27
Formal Charge0
Complexity473
Isotope Atom Count0
Defined Atom Stereocenter Count3
Undefined Atom Stereocenter Count1
Defined Bond Stereocenter Count0
Undefined Bond Stereocenter Count0
Covalently Bonded Unit Count2
4 Pharmacology and Biochemistry
4.1 MeSH Pharmacological Classification

Adjuvants, Anesthesia

Agents that are administered in association with anesthetics to increase effectiveness, improve delivery, or decrease required dosage. (See all compounds classified as Adjuvants, Anesthesia.)


Analgesics, Opioid

Compounds with activity like OPIATE ALKALOIDS, acting at OPIOID RECEPTORS. Properties include induction of ANALGESIA or NARCOSIS. (See all compounds classified as Analgesics, Opioid.)


Narcotic Antagonists

Agents inhibiting the effect of narcotics on the central nervous system. (See all compounds classified as Narcotic Antagonists.)


Narcotics

Agents that induce NARCOSIS. Narcotics include agents that cause somnolence or induced sleep (STUPOR); natural or synthetic derivatives of OPIUM or MORPHINE or any substance that has such effects. They are potent inducers of ANALGESIA and OPIOID-RELATED DISORDERS. (See all compounds classified as Narcotics.)


API Reference Price

read-more
read-more
[{"dataSource":"API Export","activeIngredients":"","year":"2021","qtr":"Q3","strtotime":1625164200,"product":"PENTAZOCINE USP","address":"ACME PLAZA, ANDHERI KURLA ROAD,ANDHERI EAST","city":"MUMBAI, MAHARASHTRA.","supplier":"SUN PHARMACEUTICAL INDUSTRIES LIMITED","supplierCountry":"INDIA","foreign_port":"KARACHI -","customer":"MEDIATE PHARMACEUTICAL PVT ","customerCountry":"PAKISTAN","quantity":"12.10","actualQuantity":"12.1","unit":"KGS","unitRateFc":"1200","totalValueFC":"14317","currency":"USD","unitRateINR":88181.818181818191,"date":"02-Jul-2021","totalValueINR":"1067000","totalValueInUsd":"14317","indian_port":"DELHI AIR","hs_no":"29333300","bill_no":"2860385","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"PAKISTAN","selfForZScoreResived":"Pharma Grade","supplierPort":"DELHI AIR","supplierAddress":"ACME PLAZA, ANDHERI KURLA ROAD,ANDHERI EAST, MUMBAI, MAHARASHTRA.","customerAddress":""},{"dataSource":"API Export","activeIngredients":"","year":"2021","qtr":"Q3","strtotime":1629916200,"product":"PENTAZOCINE B.NO.M607200020 TO M60720002 2 MF.DT.JUL.2021 EX.DT.JUN.2026 & B.NO.M 607200023 MF.DT.AUG.2021 EX.DT.JUL.2026","address":"SCO.850, SHIVALIK ENCLAVE, NAC,MANIMAJRA,","city":"CHANDIGARH.","supplier":"IND SWIFT LABORATORIES LIMITED","supplierCountry":"INDIA","foreign_port":"KARACHI -","customer":"BANK AL HABIB ","customerCountry":"PAKISTAN","quantity":"183.35","actualQuantity":"183.35","unit":"KGS","unitRateFc":"862.3","totalValueFC":"153592.9","currency":"USD","unitRateINR":62130.325879465505,"date":"26-Aug-2021","totalValueINR":"11391595.25","totalValueInUsd":"153592.9","indian_port":"DELHI AIR","hs_no":"29333300","bill_no":"4144065","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"PAKISTAN","selfForZScoreResived":"Pharma Grade","supplierPort":"DELHI AIR","supplierAddress":"SCO.850, SHIVALIK ENCLAVE, NAC,MANIMAJRA,, CHANDIGARH.","customerAddress":""},{"dataSource":"API Export","activeIngredients":"","year":"2021","qtr":"Q3","strtotime":1629916200,"product":"PENTAZOCINE HYDROCHLORIDE BATCH NO.M0200 90001 MFG.DT.AUG.2021 EXP.DT.JUL.2026","address":"SCO.850, SHIVALIK ENCLAVE, NAC,MANIMAJRA,","city":"CHANDIGARH.","supplier":"IND SWIFT LABORATORIES LIMITED","supplierCountry":"INDIA","foreign_port":"LAHORE","customer":"SAMBA BANK LTD","customerCountry":"PAKISTAN","quantity":"5.78","actualQuantity":"5.78","unit":"KGS","unitRateFc":"1267.1","totalValueFC":"7114.7","currency":"USD","unitRateINR":91294.031141868501,"date":"26-Aug-2021","totalValueINR":"527679.5","totalValueInUsd":"7114.7","indian_port":"DELHI AIR","hs_no":"29333300","bill_no":"4143222","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"PAKISTAN","selfForZScoreResived":"Pharma Grade","supplierPort":"DELHI AIR","supplierAddress":"SCO.850, SHIVALIK ENCLAVE, NAC,MANIMAJRA,, CHANDIGARH.","customerAddress":""},{"dataSource":"API Export","activeIngredients":"","year":"2021","qtr":"Q3","strtotime":1630002600,"product":"PENTAZOCINE BATCH NO.M607200020 MFG.DT.J ULY.2021 EXP.DT.JUNE.2026","address":"SCO.850, SHIVALIK ENCLAVE, NAC,MANIMAJRA,","city":"CHANDIGARH.","supplier":"IND SWIFT LABORATORIES LIMITED","supplierCountry":"INDIA","foreign_port":"ISLAMABAD - ISLAMABA","customer":"BANK AL-HABIB LIMITED,TECHNO CITY,","customerCountry":"PAKISTAN","quantity":"3.00","actualQuantity":"3","unit":"KGS","unitRateFc":"1400.3","totalValueFC":"4081.1","currency":"USD","unitRateINR":100894.66666666667,"date":"27-Aug-2021","totalValueINR":"302684","totalValueInUsd":"4081.1","indian_port":"DELHI AIR","hs_no":"29333300","bill_no":"4156076","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"PAKISTAN","selfForZScoreResived":"Pharma Grade","supplierPort":"DELHI AIR","supplierAddress":"SCO.850, SHIVALIK ENCLAVE, NAC,MANIMAJRA,, CHANDIGARH.","customerAddress":""},{"dataSource":"API Export","activeIngredients":"","year":"2022","qtr":"Q4","strtotime":1671474600,"product":"PENTAZOCINE BATCH NO. N607200041 MFG.DT.","address":"SCO.850, SHIVALIK ENCLAVE, NAC,,MA NIMAJRA,","city":"CHANDIGARH,CHANDIGARH","supplier":"IND SWIFT LABORATORIES LIMITED","supplierCountry":"INDIA","foreign_port":"ISLAMABAD - ISLAMABA","customer":"HABIB METROPOLITAN BANK ","customerCountry":"PAKISTAN","quantity":"35.00","actualQuantity":"35","unit":"KGS","unitRateFc":"800","totalValueFC":"27631.4","currency":"USD","unitRateINR":65057.142857142855,"date":"20-Dec-2022","totalValueINR":"2277000","totalValueInUsd":"27631.4","indian_port":"DELHI AIR","hs_no":"29333324","bill_no":"6292747","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"PAKISTAN","selfForZScoreResived":"Pharma Grade","supplierPort":"DELHI AIR","supplierAddress":"SCO.850, SHIVALIK ENCLAVE, NAC,,MA NIMAJRA,, CHANDIGARH,CHANDIGARH","customerAddress":""},{"dataSource":"API Export","activeIngredients":"","year":"2023","qtr":"Q3","strtotime":1693852200,"product":"PENTAZOCINE BATCH NO. O607210002 MFG.DT.AUG.2023 EXP.DT.JUL.2028","address":"SCO.850, SHIVALIK ENCLAVE, NAC,","city":"CHANDIGARH.","supplier":"IND SWIFT LABORATORIES LIMITED","supplierCountry":"INDIA","foreign_port":"LAGOS","customer":"DRUGFIELD PHARMACEUTICALS LIMITED","customerCountry":"NIGERIA","quantity":"50.00","actualQuantity":"50","unit":"KGS","unitRateFc":"1245","totalValueFC":"61540.4","currency":"USD","unitRateINR":102320,"date":"05-Sep-2023","totalValueINR":"5116000","totalValueInUsd":"61540.4","indian_port":"Delhi Air","hs_no":"29333324","bill_no":"3709232","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"NIGERIA","selfForZScoreResived":"Pharma Grade","supplierPort":"Delhi Air","supplierAddress":"SCO.850, SHIVALIK ENCLAVE, NAC,, CHANDIGARH.","customerAddress":""},{"dataSource":"API Export","activeIngredients":"","year":"2023","qtr":"Q3","strtotime":1694543400,"product":"PENTAZOCINE BATCH NO. O607210002 MFG.DT.AUG.2023 EXP.DT.JUL.2028","address":"SCO.850, SHIVALIK ENCLAVE, NAC,","city":"CHANDIGARH.","supplier":"IND SWIFT LABORATORIES LIMITED","supplierCountry":"INDIA","foreign_port":"LAGOS","customer":"DRUGFIELD PHARMACEUTICALS LIMITED","customerCountry":"NIGERIA","quantity":"50.00","actualQuantity":"50","unit":"KGS","unitRateFc":"1245","totalValueFC":"61227.6","currency":"USD","unitRateINR":101800,"date":"13-Sep-2023","totalValueINR":"5090000","totalValueInUsd":"61227.6","indian_port":"Delhi Air","hs_no":"29333324","bill_no":"3893211","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"NIGERIA","selfForZScoreResived":"Pharma Grade","supplierPort":"Delhi Air","supplierAddress":"SCO.850, SHIVALIK ENCLAVE, NAC,, CHANDIGARH.","customerAddress":""},{"dataSource":"API Export","activeIngredients":"","year":"2024","qtr":"Q1","strtotime":1709058600,"product":"PENTAZOCINE BATCH NO.O607200046 MFG.DT.DEC.2023 EXP.DT.NOV.2028","address":"SCO.850, SHIVALIK ENCLAVE, NAC,","city":"CHANDIGARH.","supplier":"IND SWIFT LABORATORIES LIMITED","supplierCountry":"INDIA","foreign_port":"DHAKA","customer":"PUBALI BANK LTD.PANTHAPATH BRANCH,","customerCountry":"BANGLADESH","quantity":"20.00","actualQuantity":"20","unit":"KGS","unitRateFc":"1000","totalValueFC":"19748","currency":"USD","unitRateINR":81996.25,"date":"28-Feb-2024","totalValueINR":"1639925","totalValueInUsd":"19748","indian_port":"Delhi Air","hs_no":"29333324","bill_no":"7905959","productDescription":"API","marketType":"LESS REGULATED MARKET","country":"BANGLADESH","selfForZScoreResived":"Pharma Grade","supplierPort":"Delhi Air","supplierAddress":"SCO.850, SHIVALIK ENCLAVE, NAC,, CHANDIGARH.","customerAddress":""}]
02-Jul-2021
28-Feb-2024
KGS
overview
Loading...

Average Price (USD/KGS)

Number of Transactions

Total Quantity (KGS)

Total Value (USD)

Quantity (KGS) & Unit rate (USD/KGS) over time

API Imports and Exports

Importing Country Total Quantity
(KGS)
Average Price
(USD/KGS)
Number of Transactions

Upgrade, download data, analyse, strategize, subscribe with us contact

Related Excipient Companies

Upload your portfolio for free, ask us

Excipients by Applications

Click here to find the perfect excipient manufacturers by their capabilities

Fillers, Diluents & Binders

read-more
read-more

Direct Compression

read-more
read-more

Disintegrants & Superdisintegrants

read-more
read-more

Lubricants & Glidants

read-more
read-more

Granulation

read-more
read-more

Thickeners and Stabilizers

read-more
read-more

Co-Processed Excipients

read-more
read-more

Coating Systems & Additives

read-more
read-more

Controlled & Modified Release

read-more
read-more

Taste Masking

read-more
read-more

Solubilizers

read-more
read-more

Film Formers & Plasticizers

read-more
read-more

Chewable & Orodispersible Aids

read-more
read-more

Parenteral

read-more
read-more

Emulsifying Agents

read-more
read-more

Topical

read-more
read-more

Surfactant & Foaming Agents

read-more
read-more

Rheology Modifiers

read-more
read-more

API Stability Enhancers

read-more
read-more

Global Sales Information

Do you need Business Intel? Ask us

Market Place

Do you need sourcing support? Ask us

REF. STANDARDS & IMPURITIES

Upload your portfolio for free, ask us

ABOUT THIS PAGE

Ask Us for Pharmaceutical Supplier and Partner
Ask Us, Find A Supplier / Partner
No Commissions, No Strings Attached, Get Connected for FREE

What are you looking for?

How can we help you?

The request can't be empty

Please read our Privacy Policy carefully

You must agree to the privacy policy

The name can't be empty
The company can't be empty.
The email can't be empty Please enter a valid email.
The mobile can't be empty